Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ DPDPE
A potent agonist selective for δ opioid receptor (EC50
MilliporeSigma™ Calbiochem™ Dipeptidylpeptidase IV Inhibitor IV, K579
The Dipeptidylpeptidase IV Inhibitor IV, K579, also referenced under CAS 440100-64-1, controls the biological activity of Dipeptidylpeptidase IV. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ Andrographolide
A bicyclic diterpenoid lactone that displays anti-viral, anti-inflammatory, anti-apoptotic, and anti-hyperglycemic properties.
MilliporeSigma™ Calbiochem™ PFKFB3 Inhibitor III, YN1
A cell-permeable, potent and competitive inhibitor of fructose-2,6-bisphosphatase 3 (PFKFB3; IC50 = 670 nM).
MilliporeSigma™ Calbiochem™ CENTA™ β-Lactamase Substrate
CENTA™ β-Lactamase Substrate, CAS 9073-60-3, is a chromogenic β-lactamase substrate for both Gram-negative and Gram-positive bacteria.
MilliporeSigma™ Calbiochem™ DAPK Inhibitor
The DAPK Inhibitor, also referenced under CAS 315694-89-4, controls the biological activity of DAPK.
MilliporeSigma™ Calbiochem™ Mifepristone
A cell-permeable synthetic steroid that acts as a potent antagonist of progesterone and glucocorticoid receptors.
MilliporeSigma™ Calbiochem™ Brk Inhibitor, Cpd 4f
A cell permeable, highly potent, and very selective inhibitor of breast tumor kinase (Brk; IC50 = 3.15 nM). Displays anti-proliferative activity against multiple breast cancer cell lines.
MilliporeSigma™ Calbiochem™ Sphingosine Kinase 1 Inhibitor II, PF-543
The Sphingosine Kinase 1 Inhibitor II, PF-543 controls the biological activity of Sphingosine Kinase 1. This small molecule/inhibitor is primarily used for Cell Structure applications.
MilliporeSigma™ Calbiochem™ Phosphatase Inhibitor Cocktail Set III
Phosphatase Inhibitor Cocktail Set III is a ready to use cocktail of four phosphatase inhibitors for broad-spectrum inhibition of both serine/threonine and protein tyrosine phosphatases.
MilliporeSigma™ Calbiochem™ Keap1-Nrf2 Interaction Probe, ML334
A cell-permeable, direct, non-covalent inhibitor of Keap1 - Nrf2 protein - protein interaction (Kd = 1 μM) that causes the dissociation of Nrf2 from keap1 in the cytosol.
MilliporeSigma™ Calbiochem™ Stauprimide
A cell-permeable ESCs (Embryonic Stem Cells) EMT (Epithelial-Mesenchymal Transition) inducer that is reported to prime/sensitize human and murine ESC cultures for much more enhanced/efficient differentiation into progenitor cells of multiple lineages.
MilliporeSigma™ Calbiochem™ Ryanodine, High Purity
Naturally occurring alkaloid that blocks the release of Ca2+ from the sarcoplasmic reticulum.
MilliporeSigma™ Calbiochem™ Estrogen Receptor Antagonist, ICI 182,780
A cell-permeable estrogen antagonist. More effective than tamoxifen in reducing estrogen receptors in breast tumor cells.